Enalapril Maleate
Kāpae
Enalapril Maleate
wehewehe
ʻO Enalapril (maleate) (MK-421 (maleate)), ka metabolite ikaika o ka enalapril, he mea hoʻohiolo i ka angiotensin-converting enzyme (ACE).
Ma Vivo
ʻO ka Enalapril (MK-421) kahi lāʻau lapaʻau e pili ana i ka angiotensin-converting enzyme (ACE) inhibitor papa o nā lāʻau lapaʻau. Hoʻopili koke ia i loko o ke ake i ka enalaprilat ma hope o ka hoʻohana waha. ʻO Enalapril (MK-421) kahi mea hoʻokūkū ikaika a hoʻokūkū o ACE, ka enzyme kuleana no ka hoʻololi ʻana o ka angiotensin I (ATI) i ka angiotensin II (ATII). Hoʻoponopono ʻo ATII i ke koko a he mea nui ia o ka ʻōnaehana renin-angiotensin-aldosterone (RAAS). Hiki ke hoʻohana ʻia ʻo Enalapril e mālama i ka hypertension koʻikoʻi a i ʻole renovascular a me nā hōʻailona congestive heart failure.
Waihona
Pauda | -20°C | 3 makahiki |
4°C | 2 makahiki | |
I ka solvent | -80°C | 6 mahina |
-20°C | 1 mahina |
ʻO ke kinona





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